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A2 ADENOSINE RECEPTOR AGONISTS

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专利名称:A2 ADENOSINE RECEPTOR AGONISTS发明人:JACOBSON, KENNETH, A.,GAO, ZHAN-GUO,ADACHI, HAYAMITSU,DOWNEY,JAMES, M.,LIU, YANPING

申请号:US2008067978申请日:20080624

公开号:WO20090060A3公开日:20090409

摘要:Disclosed are AZB adenosine receptor (AR) agonists of formula (I), in which R1,R2, R3, R4, Z, and n are defined herein. The invention also provides compositions

comprising at least one compound of formula I and methods of use thereof, for example,in the treatment of septic shock, cystic fibrosis, restenosis, erectile dysfunction,inflammation, myocardial ischemia, and reperfusion injury.

申请人:GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THESECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES,SOUTH ALABAMAMEDICAL SCIENCE FOUNDATION,JACOBSON, KENNETH, A.,GAO, ZHAN-GUO,ADACHI,HAYAMITSU,DOWNEY, JAMES, M.,LIU, YANPING

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